Regioselectivity in the biaryl coupling reactions of 1-[(1,3-benzodioxol-5-yl)methyl]-7-iodo-2,3-dihydroindole using palladium reagent

Takashi Harayama, Akihiro Hori, Hitoshi Abe, Yasuo Takeuchi

Research output: Contribution to journalArticle

10 Citations (Scopus)

Abstract

The biaryl coupling reaction of 1-[(1,3-benzodioxol-5-yl)methyl]-7-iodo-2,3-dihydroindole (1) using Pd(OAc)2 gave selectively 4,5-dihydro-7H-[1,3]dioxolo[4,5-k]pyrrolo[3,2,1-de]phenanthridine (4), which was formed by connection to a more hindered carbon, in 3.4∼4.2:1 ratios.

Original languageEnglish
Pages (from-to)385-390
Number of pages6
JournalHeterocycles
Volume67
Issue number1
DOIs
Publication statusPublished - Jan 1 2006

ASJC Scopus subject areas

  • Analytical Chemistry
  • Pharmacology
  • Organic Chemistry

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