Abstract
Tetrahydro-β-carbolines, (S)-tetrahydroharman (8a) and (S)-1-phenyltetrahydro-β-carboline (8b), were asymmetrically synthesized starting from (R)-phenylglycinol and 1-benzy1-3-(2-bromoethy)indole (1). Asymmetric synthesis of the 9-thio analogue (15) of 8a was also achieved.
Original language | English |
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Pages (from-to) | 3338-3340 |
Number of pages | 3 |
Journal | Chemical and Pharmaceutical Bulletin |
Volume | 39 |
Issue number | 12 |
DOIs | |
Publication status | Published - 1991 |
Keywords
- 3-c]pyridine phenylglycinol asymmetric synthesis
- 5]thieno[2
- carboline (S)-tetrahydroharman (S)-aryltetrahydro-β
- carboline tetrahydroberfzo[4
- tetrahydro-β
ASJC Scopus subject areas
- Chemistry(all)
- Drug Discovery