A mild Bischler–Napieralski-type cyclization of trichloromethyl carbamates for the synthesis of β -carbolinones

Seiya Hirao; Mayumi Kitamori; Tomoki Itoh; Yuusuke Chiba; Takumi Abe

doi:10.3987/COM-19-S(F)19

A mild Bischler–Napieralski-type cyclization of trichloromethyl carbamates for the synthesis of β -carbolinones

Seiya Hirao, Mayumi Kitamori, Tomoki Itoh, Yuusuke Chiba, Takumi Abe

Research output: Contribution to journal › Article › peer-review

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Abstract

– A straightforward synthesis of β-carbolinones by the Bischler–Napieralski-type cyclization of the corresponding trichloromethyl carbamates, which does not require acids, bases, oxidants, or transition-metals to promote the cyclization, has been achieved.

Original language	English
Pages (from-to)	235-250
Number of pages	16
Journal	Heterocycles
Volume	101
Issue number	1
DOIs	https://doi.org/10.3987/COM-19-S(F)19
Publication status	Published - 2020
Externally published	Yes

ASJC Scopus subject areas

Analytical Chemistry
Pharmacology
Organic Chemistry

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title = "A mild Bischler–Napieralski-type cyclization of trichloromethyl carbamates for the synthesis of β -carbolinones",

abstract = "– A straightforward synthesis of β-carbolinones by the Bischler–Napieralski-type cyclization of the corresponding trichloromethyl carbamates, which does not require acids, bases, oxidants, or transition-metals to promote the cyclization, has been achieved.",

author = "Seiya Hirao and Mayumi Kitamori and Tomoki Itoh and Yuusuke Chiba and Takumi Abe",

note = "Funding Information: This work was financially supported by JSPS (KAKENHI Grant Number 16K18849 for T.A.) as a Publisher Copyright: {\textcopyright} 2020 The Japan Institute of Heterocyclic Chemistry",

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AU - Itoh, Tomoki

AU - Chiba, Yuusuke

AU - Abe, Takumi

PY - 2020

Y1 - 2020

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A mild Bischler–Napieralski-type cyclization of trichloromethyl carbamates for the synthesis of β -carbolinones

Abstract

ASJC Scopus subject areas

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