A convenient synthesis of C(2)-substituted cephalosporins

S. Torii, H. Tanaka, N. Saitoh

Research output: Contribution to journalArticle

6 Citations (Scopus)

Abstract

Replacement of the C(2)-substituents of 2-acetoxy- or 2-methoxycephalosporin with nucleophiles was performed efficiently in dichloromethane in the presence of acid-catalysts, affording cephalosporins bearing heteroaromatic moieties, sulfenyl, and alkoxyl groups at the C(2)-position.

Original languageEnglish
Pages (from-to)2185-2186
Number of pages2
JournalBulletin of the Chemical Society of Japan
Volume56
Issue number7
Publication statusPublished - 1983

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Bearings (structural)
Nucleophiles
Methylene Chloride
Cephalosporins
Catalysts
Acids

ASJC Scopus subject areas

  • Chemistry(all)

Cite this

Torii, S., Tanaka, H., & Saitoh, N. (1983). A convenient synthesis of C(2)-substituted cephalosporins. Bulletin of the Chemical Society of Japan, 56(7), 2185-2186.

A convenient synthesis of C(2)-substituted cephalosporins. / Torii, S.; Tanaka, H.; Saitoh, N.

In: Bulletin of the Chemical Society of Japan, Vol. 56, No. 7, 1983, p. 2185-2186.

Research output: Contribution to journalArticle

Torii, S, Tanaka, H & Saitoh, N 1983, 'A convenient synthesis of C(2)-substituted cephalosporins', Bulletin of the Chemical Society of Japan, vol. 56, no. 7, pp. 2185-2186.
Torii, S. ; Tanaka, H. ; Saitoh, N. / A convenient synthesis of C(2)-substituted cephalosporins. In: Bulletin of the Chemical Society of Japan. 1983 ; Vol. 56, No. 7. pp. 2185-2186.
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